Vasu, Kamala : rechercher sur Z-Library

Campagne de collecte 15 septembre 2024 – 1 octobre 2024 C'est quoi, la collecte de fonds?

Le plus grand référentiel d'articles scientifiques au monde. 70,000,000+ d'articles gratuitement.

Campagne de collecte 15 septembre 2024 – 1 octobre 2024

Z-Library est une des plus grandes bibliothèques en ligne dans le monde, avec le stockage de plus de 17,000,000 livres et plus de 84,837,000 articles. Nous encourageons l'accès libre de chacun à la littérature. Aujourd'hui (15 septembre 2024) nous faisons un appel de fonds à tous ceux qui veulent contribuer encore plus au soutien et au développement de notre projet.

Les téléchargements SANS LIMITE sont aussi (au cours de 31 jours après la date de don) disponibles pour TOUS les utilisateurs qui soient en mesure de soutenir le projet pendant la période de collecte de fonds jusqu'au 1 octobre 2024.

C'est quoi, la collecte de fonds?En savoir plus

Livres
Articles (53)
Les plus populaires
Liste
- Liste
- Tableau

1

Gastroretentive delivery of rifampicin: In vitro mucoadhesion and in vivo gamma scintigraphy

Swati Pund, Amita Joshi, Kamala Vasu, Manish Nivsarkar, Chamanlal Shishoo

Journal:

International Journal of Pharmaceutics

Année:

2011

Langue:

english

Fichier:

PDF, 455 KB

english, 2011

2

Stability-indicating assay method for determination of actarit, its process related impurities and degradation products: Insight into stability profile and degradation pathways☆

Abiramasundari, A., Joshi, Rahul P., Jalani, Hitesh B., Sharma, Jayesh A., Pandya, Dhaivat H., Pandya, Amit N., Sudarsanam, Vasudevan, Vasu, Kamala K.

Journal:

Journal of Pharmaceutical Analysis

Année:

2014

Langue:

english

Fichier:

PDF, 1.31 MB

english, 2014

3

ChemInform Abstract: Synthesis of 1-(5-Methylisoxazole-3-yl)-5-aryl-tetrazoles and Its Pyrolysis.

Kamala K. Vasu, K. Kondal Reddy

Journal:

Année:

1999

Fichier:

PDF, 27 KB

1999

4

ChemInform Abstract: Design, Synthesis and Characterization of Novel 2-(2,4-Disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one Derivatives as Inhibitors of NF-ϰB and AP-1 Mediated Transcription Activation and as Potential Antiinflammatory Agents.

Rajan S. Giri, Hardik M. Thaker, Tony Giordano, Jill Williams, Donna Rogers, Vasudevan Sudersanam, Kamala K. Vasu

Journal:

Année:

2009

Fichier:

PDF, 25 KB

2009

5

ChemInform Abstract: A Convenient Synthesis of Di- and Trisubstituted 2-Aminoimidazoles from 1-Amidino-3-trityl-thioureas.

Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, Hitesh B. Jalani, Kamala K. Vasu, V. Sudarsanam

Journal:

Année:

2009

Fichier:

PDF, 31 KB

2009

6

ChemInform Abstract: A Convenient One-Pot Synthesis of Trisubstituted 1,3,5-Triazines Through Intermediary Amidinothioureas.

Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, Hitesh B. Jalani, V. Sudarsanam, Kamala K. Vasu

Journal:

Année:

2010

Fichier:

PDF, 38 KB

2010

7

ChemInform Abstract: A Versatile One-Pot Multicomponent Synthesis of Novel Quinazolinon-2-yl-tetrasubstituted Thiophenes.

Hitesh B. Jalani, Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, V. Sudarsanam, Kamala K. Vasu

Journal:

Année:

2011

Fichier:

PDF, 32 KB

2011

8

ChemInform Abstract: An Efficient Synthesis of 2-Aminopyrroles from Enaminone—Amidine Adduct and Phenacyl/Benzyl/Heteroalkyl-Halides.

Hitesh B. Jalani, Amit N. Pandya, Arshi B. Baraiya, Jitendra C. Kaila, Dhaivat H. Pandya, Jayesh A. Sharma, V. Sudarsanam, Kamala K. Vasu

Journal:

Année:

2012

Fichier:

PDF, 28 KB

2012

9

Design, synthesis, and pharmacological evaluation of some 2-[4-morpholino]-3-aryl-5-substituted thiophenes as novel anti-inflammatory agents: generation of a novel anti-inflammatory pharmacophore

Ajay D. Pillai, Parendu D. Rathod, Franklin P. Xavier, Kamala K. Vasu, Harish Padh, Vasudevan Sudarsanam

Journal:

Bioorganic & Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 277 KB

english, 2004

10

QSAR studies on some thiophene analogs as anti-inflammatory agents: enhancement of activity by electronic parameters and its utilization for chemical lead optimization

Ajay D. Pillai, Shubha Rani, Parendu D. Rathod, Franklin P. Xavier, Kamala K. Vasu, Harish Padh, Vasudevan Sudarsanam

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 313 KB

english, 2005

11

Tetra substituted thiophenes as anti-inflammatory agents: Exploitation of analogue-based drug design

Ajay D. Pillai, Parendu D. Rathod, Franklin P. Xavier, Harish Padh, Vasudevan Sudarsanam, Kamala K.Vasu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 172 KB

english, 2005

12

Multivariate optimization of formulation and process variables influencing physico-mechanical characteristics of site-specific release isoniazid pellets

Swati Pund, Amita Joshi, Kamala Vasu, Manish Nivsarkar, Chamanlal Shishoo

Journal:

International Journal of Pharmaceutics

Année:

2010

Langue:

english

Fichier:

PDF, 564 KB

english, 2010

13

2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists

Anja B. Scheiff, Swapnil G. Yerande, Ali El-Tayeb, Wenjin Li, Gajanan S. Inamdar, Kamala K. Vasu, Vasudevan Sudarsanam, Christa E. Müller

Journal:

Bioorganic & Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 697 KB

english, 2010

14

Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents

Khurshid I. Molvi, Kamala K. Vasu, Swapnil G. Yerande, Vasudevan Sudarsanam, Navedul Haque

Journal:

European Journal of Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 228 KB

english, 2007

15

2-Amino-5-thiazolyl motif: A novel scaffold for designing anti-inflammatory agents of diverse structures

P.X. Franklin, Ajay D. Pillai, Parendu D. Rathod, Swapnil Yerande, Manish Nivsarkar, Harish Padh, Kamala K. Vasu, V. Sudarsanam

Journal:

European Journal of Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 237 KB

english, 2008

16

Design, synthesis and characterization of novel 2-(2,4-disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one derivatives as inhibitors of NF-κB and AP-1 mediated transcription activation and as potential anti-inflammatory agents

Rajan S. Giri, Hardik M. Thaker, Tony Giordano, Jill Williams, Donna Rogers, Vasudevan Sudersanam, Kamala K. Vasu

Journal:

European Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 291 KB

english, 2009

17

Corrigendum to “Design, synthesis and characterization of novel 2-(2,4-disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one derivatives as inhibitors of NF-κB and AP-1 mediated transcription activation and as potential anti-inflammatory agents” [Eur J Med Chem 44 (2009) 2184–2189]

Rajan S. Giri, Hardik M. Thaker, Tony Giordano, Jill Williams, Donna Rogers, Vasudevan Sudersanam, Kamala K. Vasu

Journal:

European Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 78 KB

english, 2009

18

A facile synthesis of structurally novel 1-aryl-2-arylamino-4-alkyl/phenyl-5-aroyl-1H-imidazoles from amidinothioureas

Jitendra C. Kaila, Arshi B. Baraiya, Kamala K. Vasu, V. Sudarsanam

Journal:

Tetrahedron Letters

Année:

2008

Langue:

english

Fichier:

PDF, 172 KB

english, 2008

19

A convenient synthesis of di- and trisubstituted 2-aminoimidazoles from 1-amidino-3-trityl-thioureas

Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, Hitesh B. Jalani, Kamala K. Vasu, V. Sudarsanam

Journal:

Tetrahedron Letters

Année:

2009

Langue:

english

Fichier:

PDF, 388 KB

english, 2009

20

A convenient one-pot synthesis of trisubstituted 1,3,5-triazines through intermediary amidinothioureas

Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, Hitesh B. Jalani, V. Sudarsanam, Kamala K. Vasu

Journal:

Tetrahedron Letters

Année:

2010

Langue:

english

Fichier:

PDF, 2.52 MB

english, 2010

21

A versatile one-pot multicomponent synthesis of novel quinazolinon-2-yl-tetrasubstituted thiophenes

Hitesh B. Jalani, Jitendra C. Kaila, Arshi B. Baraiya, Amit N. Pandya, V. Sudarsanam, Kamala K. Vasu

Journal:

Tetrahedron Letters

Année:

2010

Langue:

english

Fichier:

PDF, 395 KB

english, 2010

22

Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-кB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents

Rajan S. Giri, Hardik M. Thaker, Tony Giordano, Jill Williams, Donna Rogers, Kamala K. Vasu, Vasudevan Sudarsanam

Journal:

Bioorganic & Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 1.17 MB

english, 2010

23

Synthesis and evaluation of quinazolinone derivatives as inhibitors of NF-κB, AP-1 mediated transcription and eIF-4E mediated translational activation: Inhibitors of multi-pathways involve in cancer

Rajan S. Giri, Hardik M. Thaker, Tony Giordano, Bing Chen, Sam Nuthalapaty, Kamala K. Vasu, Vasudevan Sudarsanam

Journal:

European Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 437 KB

english, 2010

24

An efficient synthesis of 2-aminopyrroles from enaminone–amidine adduct and phenacyl/benzyl/heteroalkyl-halides

Hitesh B. Jalani, Amit N. Pandya, Arshi B. Baraiya, Jitendra C. Kaila, Dhaivat H. Pandya, Jayesh A. Sharma, V. Sudarsanam, Kamala K. Vasu

Journal:

Tetrahedron Letters

Année:

2011

Langue:

english

Fichier:

PDF, 2.58 MB

english, 2011

25

An efficient, greener, and solvent-free one-pot multicomponent synthesis of 3-substituted quinazolin-4(3H)ones and thienopyrimidin-4(3H)ones

Hitesh B. Jalani, Amit N. Pandya, Dhaivat H. Pandya, Jayesh A. Sharma, V. Sudarsanam, Kamala K. Vasu

Journal:

Tetrahedron Letters

Année:

2012

Langue:

english

Fichier:

PDF, 1.09 MB

english, 2012

26

Design, synthesis, and SAR studies of some 5-aliphatic oximino esters of thiophene as potential anti-inflammatory leads: comparative biological activity profile of aliphatic oximes vs aromatic oximes

Ajay D Pillai, Parendu D Rathod, P.X Franklin, Harish Padh, Kamala K Vasu, V Sudarsanam

Journal:

Biochemical and Biophysical Research Communications

Année:

2004

Langue:

english

Fichier:

PDF, 259 KB

english, 2004

27

Dissolution test for site-specific release isoniazid pellets in USP apparatus 3 (reciprocating cylinder): Optimization using response surface methodology

Amita Joshi, Swati Pund, Manish Nivsarkar, Kamala Vasu, Chamanlal Shishoo

Journal:

European Journal of Pharmaceutics and Biopharmaceutics

Année:

2008

Langue:

english

Fichier:

PDF, 624 KB

english, 2008

28

Novel drug designing approach for dual inhibitors as anti-inflammatory agents: implication of pyridine template

Ajay D Pillai, Parendu D Rathod, Franklin P.X, Manoj Patel, Manish Nivsarkar, Kamala K Vasu, Harish Padh, Vasudevan Sudarsanam

Journal:

Biochemical and Biophysical Research Communications

Année:

2003

Langue:

english

Fichier:

PDF, 106 KB

english, 2003

29

ChemInform Abstract: An Efficient, Greener, and Solvent-Free One-Pot Multicomponent Synthesis of 3-Substituted Quinazolin-4(3H)ones and Thienopyrimidin-4(3H)ones.

Jalani, Hitesh B., Pandya, Amit N., Pandya, Dhaivat H., Sharma, Jayesh A., Sudarsanam, V., Vasu, Kamala K.

Journal:

Année:

2012

Fichier:

PDF, 27 KB

2012

30

A concise, greener, solvent-free novel one-pot synthesis of trisubstituted thiophenes

Jalani, Hitesh B., Pandya, Amit N., Pandya, Dhaivat H., Sharma, Jayesh A., Sudarsanam, V., Vasu, Kamala K.

Journal:

Tetrahedron Letters

Année:

2012

Langue:

english

Fichier:

PDF, 1.30 MB

english, 2012

31

An efficient one-pot synthesis of functionally diverse 2-aminothiazoles from isothiocyanates, amidines/guanidines and halomethylenes

Jalani, Hitesh B., Pandya, Amit N., Pandya, Dhaivat H., Sharma, Jayesh A., Sudarsanam, V., Vasu, Kamala K.

Journal:

Tetrahedron Letters

Année:

2013

Langue:

english

Fichier:

PDF, 507 KB

english, 2013

32

3D-QSAR studies for the binding affinity toward (R, S)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)-propionic acid receptor

Sharma, Ritesh, Thakar, Hardik, Vasu, Kamala, Chaturvedi, Subhash

Journal:

Acta Pharmaceutica

Année:

2008

Langue:

english

Fichier:

PDF, 114 KB

english, 2008

33

Role of lipid-based excipients and their composition on the bioavailability of antiretroviral self-emulsifying formulations

Chudasama, Arpan, Patel, Vineetkumar, Nivsarkar, Manish, Vasu, Kamala, Shishoo, Chamanlal

Journal:

Année:

2015

Langue:

english

Fichier:

PDF, 346 KB

english, 2015

34

New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1,3-thiazol-2-yl] benzamides and furamides

Inamdar, Gajanan S., Pandya, Amit N., Thakar, Hardik M., Sudarsanam, Vasudevan, Kachler, Sonja, Sabbadin, Davide, Moro, Stefano, Klotz, Karl-Norbert, Vasu, Kamala K.

Journal:

European Journal of Medicinal Chemistry

Année:

2013

Langue:

english

Fichier:

PDF, 1.82 MB

english, 2013

35

Pair wise binding affinity: 3D QSAR studies on a set of triazolo [1, 5-a] quinoxalines as antagonists of AMPA and KA receptors

Sharma, Ritesh N., Thakar, Hardik M., Vasu, Kamala K., Chaturvedi, Subhash C., Pancholi, Shyam S.

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 920 KB

english, 2009

36

Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: An analogue-based drug design approach

Sharma, Ritesh N., Xavier, Franklin P., Vasu, Kamala K., Chaturvedi, Subhash C., Pancholi, Shyam S.

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 230 KB

english, 2009

37

Push-pull osmotic pump for zero order delivery of lithium carbonate: Development and in vitro characterization

Patel, Vineetkumar, Chudasama, Arpan, Nivsarkar, Manish, Vasu, Kamala, Shishoo, Chamanlal

Journal:

Pharmaceutical Development and Technology

Année:

2012

Langue:

english

Fichier:

PDF, 1.21 MB

english, 2012

38

Implication of novel bis-imidazopyridines for management of Alzheimer's disease and establishment of its role on protein phosphatase 2A activity in brain

Parekh, Kauntay D., Dash, Ranjeet Prasad, Pandya, Amit N., Vasu, Kamala K., Nivsarkar, Manish

Journal:

Journal of Pharmacy and Pharmacology

Année:

2013

Langue:

english

Fichier:

PDF, 784 KB

english, 2013

39

Novel thiazole–thiophene conjugates as adenosine receptor antagonists: Synthesis, biological evaluation and docking studies

Pandya, Dhaivat H., Sharma, Jayesh A., Jalani, Hitesh B., Pandya, Amit N., Sudarsanam, V., Kachler, Sonja, Klotz, Karl Norbert, Vasu, Kamala K.

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2015

Langue:

english

Fichier:

PDF, 508 KB

english, 2015

40

Development of self emulsifying drug delivery system of itraconazole for oral delivery: formulation and pharmacokinetic consideration

Chudasama, Arpan, Shah, Brijesh, Patel, Vineetkumar, Nivsarkar, Manish, Vasu, Kamala, Shishoo, Chamanlal

Journal:

Journal of Pharmaceutical Investigation

Année:

2015

Langue:

english

Fichier:

PDF, 655 KB

english, 2015

41

ChemInform Abstract: A Diversified Assembly of 1,2,4-Oxadiazol-3-amines: Metallic Thiophile Catalyzed Chemoselective One-Pot Reaction of Aryl Isothiocyanates, Amidines/Guanidines, and Hydroxylamine.

Jalani, Hitesh B., Sudarsanam, V., Vasu, Kamala K.

Journal:

Année:

2013

Fichier:

PDF, 28 KB

2013

42

Synthesis of 1-(5-Methylisoxazole-3-yl)-5-Aryl-Tetrazoles and its Pyrolysis

Vasu, Kamala K., Reddy, K. Kondal

Journal:

Synthetic Communications

Année:

1999

Langue:

english

Fichier:

PDF, 316 KB

english, 1999

43

Characterization of Degradation Products of Bambuterol Using LCMS-QTOF and NMR

Abiramasundari, Arumugam, Vasudevan, Sudarsanam, vasu, kamala kunju

Journal:

Analytical Methods

Année:

2015

Langue:

english

Fichier:

PDF, 2.86 MB

english, 2015

44

Impact of Ternary Solvent System in Stability-Indicating Assay Method of Bambuterol: Design of Experiments Approach

Abiramasundari, A., Joshi, Amita, Joshi, Rahul, Pandya, Dhaivat, Sharma, Jayesh, Sudarsanam, V., Vasu, Kamala K.

Journal:

Journal of Chromatographic Science

Année:

2015

Langue:

english

Fichier:

PDF, 773 KB

english, 2015

45

Design, synthesis and biological evaluation of novel pyrazolo-pyrimidinones as DPP-IV inhibitors in diabetes

Sagar, Sneha R., Agarwal, Jessica K., Pandya, Dhaivat H., Dash, Ranjeet Prasad, Nivsarkar, Manish, Vasu, Kamala K.

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2015

Langue:

english

Fichier:

PDF, 1.14 MB

english, 2015

46

A Diversified Assembly of 1,2,4-Oxadiazol-3-amines: Metallic Thiophile Catalyzed Chemoselective One-Pot Reaction of Aryl Isothiocyanates, Amidines/Guanidines, and Hydroxylamine

Jalani, Hitesh, Sudarsanam, V., Vasu, Kamala

Journal:

Année:

2012

Langue:

english

Fichier:

PDF, 248 KB

english, 2012

47

ChemInform Abstract: A Concise, Greener, Solvent-Free Novel One-Pot Synthesis of Trisubstituted Thiophenes.

Jalani, Hitesh B., Pandya, Amit N., Pandya, Dhaivat H., Sharma, Javesh A., Sudarsanam, V., Vasu, Kamala K.

Journal:

Année:

2013

Fichier:

PDF, 25 KB

2013

48

Identification of dual kinase inhibitors of CK2 and GSK3β: combined qualitative and quantitative pharmacophore modeling approach

Pardhi, Triveni, Vasu, Kamala

Journal:

Journal of Biomolecular Structure and Dynamics

Année:

2017

Langue:

english

Fichier:

PDF, 1.55 MB

english, 2017

49

Imidazo[1,2- a ]pyridines linked with thiazoles/thiophene motif through keto spacer as potential cytotoxic agents and NF-κB inhibitors

Vasu, Kamala K., Digwal, Chander Singh, Pandya, Amit N., Pandya, Dhaivat H., Sharma, Jayesh A., Patel, Sneha, Agarwal, Milee

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2017

Langue:

english

Fichier:

PDF, 549 KB

english, 2017

50

Discovery of 2-aminoimidazole and 2-amino imidazolyl-thiazoles as non-xanthine human adenosine A 3 receptor antagonists: SAR and molecularmodeling studies

Pandya, Amit N., Baraiya, Arshi B., Jalani, Hitesh B., Pandya, Dhaivat, Kaila, Jitendra C., Kachler, Sonja, Salmaso, Veronica, Moro, Stefano, Klotz, Karl-Norbert, Vasu, Kamala K.

Journal:

Année:

2018

Langue:

english

Fichier:

PDF, 2.70 MB

english, 2018